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(54) DIACYLHYDRAZIN-LIGANDEN ZUR MODULATION DER EXPRESSION
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REZEPTORKOMPLEX
(72) HORMANN, Robert, Eugene, Melrose Park, PA 19027, 7413 Richards Road
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(72) TICE, Colin, M., Elkins Park, PA 19027, 1211 Stratford Avenue (US)
(72) CHORTYK, Orestes, Thompson Station, TN 37179, 3025 Liverpool Drive (US)
(72) SMITH, Howard, Landsdowne, PA 19050, 82 East Greenwood Avenue (US)
(72) METEYER, Thomas, Lansdale, PA 19446, 427 Country Club Drive (US)
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(73) Les Laboratoires Servier, 92284 Suresnes Cedex, 35, rue de Verdun (FR)
(54) Verfahren zur industriellen Herstellung von Strontiumranelat und seinen
Hydraten
(72) Vaysse-Ludot, Lucile, 76490 Saint Wandrille Rançon, 150, route de Rançon
(FR)
(72) Lecouve, Jean-Pierre, 76600 Le Havre, 93, rue du Docteur Vigné (FR)
(72) Langlois, Pascal, 76210 Saint Jean de la Neuville, 3, allée du Bassin (FR)
(30) FR 2002 09 24 0211763
(73) ONO PHARMACEUTICAL CO., LTD., Osaka-shi, Osaka 541-8526, 1-5,
Doshomachi 2-chome Chuo-ku (JP)
(54) STICKSTOFFHALTIGE HETEROCYCLISCHE VERBINDUNG UND
PHARMAZEUTISCHE ANWENDUNG DAVON
(72) NAKAI, Hisao, Osaka 618-8585, c/o ONO PHARMACEUTICAL CO., LTD., 1-
1, Sakurai 3-c home, Shimamoto-cho, Mishima-gun (JP)
(72) YAMAMOTO, Shingo, Osaka 618-8585, c/o ONO PHARMACEUTICAL CO.,
LTD., 1-1, Sakurai 3-c home, Shimamoto-cho, Mishima-gun (JP)
(72) NAKATANI, Shingo, Osaka 618-8585, c/o ONO PHARMACEUTICAL CO.,
LTD., 1-1, Sakurai 3-c home, Shimamoto-cho, Mishima-gun (JP)
(72) HIROSAKI, Tomomi, Osaka 618-8585, c/o ONO PHARMACEUTICAL CO.,
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(73) Bayer Intellectual Property GmbH, 40789 Monheim, Alfred-Nobel-Strasse 10
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(54) FLUORIERTE 2,6-DIALKYL-3,5-DICYANO-4-(1H-INDAZOL-5-YL)-1,4-
DIHYDROPYRIDINE UND VERWENDUNGSVERFAHREN DAFÜR
(72) MICHELS, Martin, 51109 Köln, Am Klausenberg 55 (DE)
(72) FOLLMANN, Markus, 42489 Wülfrath, Ringstr. 61 (DE)
(72) VAKALOPOULOS, Alexandros, 40721 Hilden, Heinrich-Heine-Str. 79a (DE)
(72) ZIMMERMANN, Katja, 40489 Düsseldorf, Bockumerstr. 370 (DE)
(72) TEUSCH, Nicole, 42489 Wülfrath, Ringstr. 61 (DE)
(72) LOBELL, Mario, 42113 Wuppertal, Am Eigenbach 16 (DE)
(72) ENGEL, Karen, 42327 Wuppertal, Goethestr. 55 (DE)
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(73) AbbVie Deutschland GmbH & Co KG, 65205 Wiesbaden, Max-Planck-Ring 2a
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(73) AbbVie Inc., North Chicago, IL 60064, 1 North Waukegan Road (US)
(54) CARBOXAMIDVERBINDUNGEN UND IHRE VERWENDUNG ALS CALPAIN-
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(72) KLING, Andreas, 67061 Ludwigshafen, c/o Abbott GmbH&Co. KG Knollstr. 50
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(72) JANTOS, Katja, 67061 Ludwigshafen, c/o Abbott GmbH&Co. KG Knollstr. 50
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(72) MACK, Helmut, 67061 Ludwigshafen, c/o Abbott GmbH&Co. KG Knollstr. 50
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(72) MÖLLER, Achim, 67061 Ludwigshafen, c/o Abbott GmbH&Co. KG Knollstr. 50
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(72) HORNBERGER, Wilfried, 67061 Ludwigshafen, c/o Abbott GmbH&Co. KG
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(72) BACKFISCH, Gisela, 67061 Ludwigshafen, c/o Abbott GmbH&Co. KG
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(72) LAO, Yanbin, Illinois 60064-6050, c/o Abbott Laboratories 100 Abbott Park
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(72) NIJSEN, Marjoleen, Illinois 60064-6050, c/o Abbott Laboratories 100 Abbott
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(73) Janssen R&D Ireland, Eastgate, Little Island, County Cork, Eastgate Village
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(54) MACROCYCLISCHE INHIBITOREN DES HEPATITIS-C-VIRUS
(72) RABOISSON, Pierre Jean-Marie Bernard, 1331 Rosieres, Rue Jolie 3 (BE)
(72) DE KOCK, Herman Augustinus, 2370 Arendonk, Wolfseind 10 (BE)
(72) MC GOWAN, David Craig, 1150 Brussel, De Biolleylaan 80 (BE)
(72) VAN DE VREKEN, Wim, 9120 Haasdonk, Willem Van Doornyckstraat 49 (BE)
(72) HU, Lili, 2800 Mechelen, Vrouw van Mechelenstraat 28 (BE)
(72) TAHRI, Abdellah, 1070 Anderlecht, Rue Maurice Albert Raskin 30 (BE)
(72) VENDEVILLE, Sandrine Marie Helene, 1150 Woluwe-Saint-Pierre, Rue du
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(30) EP 2006 11 17 06124359
(73) Academia Sinica, Taipei 115, 128, Sec. 2 Academia Sinica Road Nan-Kang
(TW)
(54) Fluoreszierende Carbazolverbindungen zur Krebsdiagnose
(72) Chang, Ta-Chau, Taipei , IAMS Academia Sinica P.O. Box 23-166 (TW)
(72) Cho, Chih-Chien, Sinjhuang City Taipei County 242, 5F, No. 13, Fong 1 st Ln.,
Fongian St. (TW)
(72) Chang, Cheng-Chung, Taichung , Graduate Institute of Biomedical
Engineering National Chung-Hsing University 250, Kuo Kuang Road (TW)
(72) Kang, Chi-Chih, Yongkang City Tainan County 710, No. 10, Ln.33, Yongpu St.
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(72) Wang, Zi-Fu, Linkou Township Taipei County 244, 11F-2, No.9, Ln.11 Liyuan
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(73) AstraZeneca AB, 151 85 Södertälje (SE)
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(72) ALCARAZ, Marie-Lyne, Loughborough Leicestershire LE11 5RH,
AstraZeneca R&D Charnwood Bakewell Road (GB)
(72) BRIGGNER, Lars-Erik, SE - 431 83 Mölndal, AstraZeneca R&D Molndal (SE)
(72) KLINGSTEDT, Per, Tomas, S-221 87 Lund, AstraZeneca R&D Lund (SE)
(72) LÖNN, Hans, Roland, SE - 431 83 Mölndal, AstraZeneca R&D Molndal (SE)
(72) NICKLASSON, Helena, SE - 151 85 Sodertalje, C/o AstraZeneca Intellectual
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(72) NIXON, Robert, Anthony, Loughborough Leicestershire LE11 5RH,
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(72) WATTS, Andrew, James, Macclesfield, Cheshire, SK10 4TG, c/o AstraZeneca
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(73) J. Uriach y Compania S.A., 08184 Palau-solità i Plegamans (Barcelona), Av.
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(54) RUPATADINderivat ALS ANTIHISTAMINIKUM
(72) CARCELLER GONZÁLEZ, Elena, E-08190 Sant Cugat del Vallès -
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(73) Merck Sharp & Dohme Corp., Rahway, NJ 07065-0907, 126 East Lincoln
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(54) THROMBINREZEPTORANTAGONISTEN
(72) CHACKALAMANNIL, Samuel, Califon, NJ 07830, 17 Windy Heights Road
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(72) CHELLIAH, Mariappan, V., Edison, NJ 08820, 56 Portland Street (US)
(72) XIA, Yan, Edison, NJ 08820, 66 Tower Road (US)
(30) US 2003 09 25 671216
(73) The Board of Trustees of the Leland Stanford Junior University, Palo Alto, CA
94306-1106, 1705 El Camino Real (US)
(54) MODULATOREN DER ALDEHYDDEHYDROGENASE-AKTIVITÄT UND
ANWENDUNGSVERFAHREN FÜR DIESE
(72) YANG, Wenjin, Foster City California 94404, 383 Bodega Street (US)
(72) CHEN, Che-Hong, Fremont California 94539, 45696 Bridgeport Drive (US)
(72) MOCHLY-ROSEN, Daria, Menlo Park California 94025, 825 Harvard Avenue
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Österreichisches Patentblatt 111. Jahrgang Nummer 4, Seite 1260
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